ent-Verticilide B1 Inhibits Type 2 Ryanodine Receptor Channels and is Antiarrhythmic in Casq2-/- MiceS
- Creator: Gochman, Aaron , Do, Tri Q. , Cornea, Razvan L. , Laver, Derek R. , Johnston, Jeffrey N. , Knollmann, Bjorn C. , Kim, Kyungsoo , Schwarz, Jacob A. , Thorpe, Madelaine P. , Blackwell, Daniel J. , Ritschel, Paxton A. , Smith, Abigail N. , Rebbeck, Robyn T. , Akers, Wendell S.
- Resource Type: journal article
- Date: 2024
A bivalent remipede toxin promotes calcium release via ryanodine receptor activation
- Creator: Maxwell, Michael J. , Thekkedam, Chris , Launikonis, Bradley S. , Dulhunty, Angela , Undheim, Eivind A. B. , Mobli, Mehdi , Lamboley, Cedric , Chin, Yanni K.-Y. , Crawford, Theo , Smith, Jennifer J. , Liu, Junyu , Jia, Xinying , Vetter, Irina , Laver, Derek R.
- Resource Type: journal article
- Date: 2023
Dantrolene inhibition of ryanodine channels (RyR2) in artificial lipid bilayers depends on FKBP12.6
- Creator: Walweel, Kafa , Beard, Nicole , van Helden, Dirk F. , Laver, Derek R.
- Resource Type: journal article
- Date: 2023
RYR2 channel inhibition is the principal mechanism of flecainide action in CPVT
- Creator: Kryshtal, Dmytro O. , Blackwell, Daniel J. , Egly, Christian L. , Smith, Abigail N. , Batiste, Suzanne M. , Johnston, Jeffrey N. , Laver, Derek R. , Knollmann, Bjorn C.
- Resource Type: journal article
- Date: 2021
Calmodulin inhibition of human RyR2 channels requires phosphorylation of RyR2-S2808 or RyR2-S2814
- Creator: Walweel, Kafa , Gomez-Hurtado, Nieves , Laver, Derek R. , Rebbeck, Robyn T. , Oo, Ye Wint , Beard, Nicole A. , Molenaar, Peter , dos Remedios, Chris , van Helden, Dirk F. , Cornea, Razvan L. , Knollmann, Björn C.
- Resource Type: journal article
- Date: 2019
Mammalian TRP on channels are insensitive to membrane stretch
- Creator: Nikolaev, Yury A. , Cox, Charles D. , Ridone, Pietro , Rohde, Paul R. , Cordero-Morales, Julio F. , Vasquez, Valeria , Laver, Derek R. , Martinac, Boris
- Resource Type: journal article
- Date: 2019
Secretoneurin is an endogenous calcium/calmodulin-dependent protein kinase II inhibitor that attenuates Ca2+-dependent arrhythmia
- Creator: Ottesen, Anett H. , Carlson, Catherine R. , Lunde, Marianne , Hoff, Jon Erik , Godang, Kristin , Sjaastad, Ivar , Pettilä, Ville , Stridsberg, Mats , Lehnart, Stephan E. , Edwards, Andrew G. , Lunde, Ida G. , Omland, Torbjørn , Eken, Olav Søvik , Stokke, Mathis K. , Christensen, Geir , Røsjø, Helge , Louch, William E. , Sadredini, Mani , Myhre, Peder L. , Shen, Xin , Dalhus, Bjørn , Laver, Derek R. , Lunde, Per Kristian , Kurola, Jouni
- Resource Type: journal article
- Date: 2019
Regulation of the RyR channel gating by Ca²⁺ and Mg²⁺
- Creator: Laver, Derek R.
- Resource Type: journal article
- Date: 2018
Cardiac calcium release channel (ryanodine receptor 2) regulation by halogenated anesthetics
- Creator: Laver, Derek R. , Attia, John , Oldmeadow, Christopher , Quail, Anthony W.
- Resource Type: journal article
- Date: 2017
Nerve-induced responses of mouse vaginal smooth muscle
- Creator: van Helden, Dirk F. , Kamiya, Ayumi , Kelsey, Sam , Laver, Derek R. , Jobling, Phillip , Mitsui, Retsu , Hashitani, Hikaru
- Resource Type: journal article
- Date: 2017
The emerging role of calmodulin regulation of RyR2 in controlling heart rhythm, the progression of heart failure and the antiarrhythmic action of dantrolene
- Creator: Walweel, Kafa , Oo, Ye Win , Laver, Derek R.
- Resource Type: journal article
- Date: 2017
A parallel modelling algorithm for simulating calcium release in cells
- Creator: Stoddard, Jeremy G. , Welsh, James S. , Laver, Derek R.
- Resource Type: conference paper
- Date: 2016
Essential role of calmodulin in RyR inhibition by dantrolene
- Creator: Oo, Ye Win , Gomez-Hurtado, Nieves , Walweel, Kafa , van Helden, Dirk F. , Imtiaz, Mohammad S. , Knollmann, Bjorn C. , Laver, Derek R.
- Resource Type: journal article
- Date: 2015
Polarized and persistent Ca²⁺ plumes define loci for formation of wall ingrowth papillae in transfer cells
- Creator: Zhang, Hui-Ming , Imtiaz, Mohammad S. , Laver, Derek R. , McCurdy, David W. , Offler, Christina E. , van Helden, Dirk F. , Patrick, John W.
- Resource Type: journal article
- Date: 2015
Single mechanically-gated cation channel currents can trigger action potentials in neocortical and hippocampal pyramidal neurons
- Creator: Nikolaev, Yury A. , Dosen, Peter J. , Laver, Derek R. , van Helden, Dirk F. , Hamill, Owen P.
- Resource Type: journal article
- Date: 2015
Differences in the regulation of RyR2 from human, sheep, and rat by Ca²⁺ and Mg²⁺ in the cytoplasm and in the lumen of the sarcoplasmic reticulum
- Creator: Walweel, Kafa , Li, Jiao , Molenaar, Peter , Imtiaz, Mohammad S. , Quail, Anthony , dos Remedios, Chris G. , Beard, Nicole A. , Dulhunty, Angela F. , van Helden, Dirk F. , Laver, Derek R.
- Resource Type: journal article
- Date: 2014
Pharmacological approaches that slow lymphatic flow as a snakebite first aid
- Creator: van Helden, Dirk F. , Thomas, Paul A. , Dosen, Peter J. , Imtiaz, Mohammad S. , Laver, Derek R. , Isbister, Geoffrey K.
- Resource Type: journal article
- Date: 2014
Beta-adrenergic stimulation increases RyR2 activity via intracellular Ca²⁺ and Mg²⁺ regulation
- Creator: Li, Jiao , Imtiaz, Mohammad S. , Beard, Nicole A. , Dulhunty, Angela F. , Thorn, Rick , van Helden Dirk F. , Laver, Derek R.
- Resource Type: journal article
- Date: 2013
Extraction of sub-microscopic Ca fluxes from blurred and noisy fluorescent indicator images with a detailed model fitting approach
- Creator: Kong, Cherrie H. T. , Laver, Derek R. , Cannell, Mark B.
- Resource Type: journal article
- Date: 2013
Selective modulation of different GABAA receptor isoforms by diazepam and etomidate in hippocampal neurons
- Creator: Seymour, Victoria A. L. , Curmi, John P. , Howitt, Susan M. , Casarotto, Marco G. , Laver, Derek R. , Tierney, M. Louise
- Resource Type: journal article
- Date: 2012